Author(s) Ayothiraman, R.; Rangaswamy, S.; Maity, P.; Simmons, E.M.; Beutner, G.L.; Janey, J.; Treitler, D.S.; Eastgate, M.D.; Vaidyanathan, R.
Journal J Org Chem
Date Published 2017 Jul 05
Abstract

Zinc salts have been shown to promote the Buchwald-Hartwig coupling of azaindoles and azaindazoles with heteroaryl chlorides to provide the corresponding 1-aryl-1H-azaindoles and 1-aryl-1H-azaindazoles. The substrate scope and mechanistic aspects of this reaction were explored.

DOI 10.1021/acs.joc.7b01101
ISSN 1520-6904
Citation Ayothiraman R, Rangaswamy S, Maity P, Simmons EM, Beutner GL, Janey J, et al. Zinc Acetate-Promoted Buchwald-Hartwig Couplings of Heteroaromatic Amines. J Org Chem. 2017.

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