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Enzymes & Inhibitors page banner

Enzymes & Inhibitors

(

(8S,10S)-10-(((2R,4S,5S,6S)-4-Amino-5-hydroxy-6-methyltetrahydro-2H-pyran-2-yl)oxy)-6,8,11-trihydroxy-8-(2-hydroxyacetyl)-1-methoxy-7,8,9,10-tetrahydrotetracene-5,12-dione hydrochloride
(R)-( )-Etomoxir Sodium
(R)-Ethyl 2-(6-(4-chlorophenoxy)hexyl)oxirane-2-carboxylate
(S)-(2,3-Dimethoxyphenyl)(1-(4-fluorophenethyl)piperidin-4-yl)methanol
(Z)-3-(3-(3,5-Bis(trifluoromethyl)phenyl)-1H-1,2,4-triazol-1-yl)-N'-(pyrazin-2-yl)acrylohydrazide

1

1-Benzyl-3-hexylguanidine Hydrochloride

2

2'-O-methyl-P-thiouridylyl-(3'-5')-2'-deoxy-Adenosine

3

3-(1H-Indol-5-yl)-5-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-1H-pyrrolo[2,3-b]pyridine
3-Acetylphenyl ethyl(methyl)carbamate
3-Isopropyl-5-(4-(((6-(4-(methylsulfonyl)phenyl)pyridin-3-yl)oxy)methyl)piperidin-1-yl)-1,2,4-oxadiazole

4

4-(5-((3-Benzyl-4-oxo-2-thioxothiazolidin-5-ylidene)methyl)furan-2-yl)benzoic acid
4-Amino-8-(2,5-dimethoxyphenyl)-N-propylcinnoline-3-carboxamide

5

5-((5-Chloro-1H-pyrrolo[2,3-b]pyridin-3-yl)methyl)-N-(4-(trifluoromethyl)benzyl)pyridin-2-amine

8

8-Nitrotryptanthrin

A

A 438079 hydrochloride
A-1210477
A-205804
A939572
ABBV-744
ABT-263
ABX464
Acetoacetyl Coenzyme A Lithium Salt
AF-64394
AG-120
AGI-6780
Alisertib
AMG-337
Amiselimod Hydrochloride
AR-42
ARS-853
AS-1842856
As-601245
ASP 9521
Asunaprevir
AT7519
AT9283
Ax20017
AZD 2098
AZD 3241
AZD 4635
AZD 7986
AZD3965
AZD5153 6-Hydroxy-2-Naphthoic Acid
AZD5438
AZD7545
AZD7762
AZD9496
Azeliragon

B

B-Raf inhibitor 1
Balicatib
Balovaptan
BAY-598
BGB324
BIX-01294
BIX-02188(Random Configuration)
BLU9931
BMS-265246
BMS-3
BMS-986020
BRL-15572 Free
BS-181 HCl
BV-6 free
BX795

c

c-Met inhibitor 1
cGAMP

C

C188-9
CC-115
CC-220
CCT-245737
Cephalosporin C zinc salt
CHIR-99021
CID-16020046
Cilengitide
CK-636
CNX-774
CP21R7
Cruzain-IN-1
CTX-0294885
CU-CPT-9b

D

D-64131
Danirixin
DAPTA
Dimethoxycurcumin
DSR-6434

E

E-6446 Dihydrochloride
E7046
ENOblock
Entecavir Monohydrate
EPZ-5676
EPZ004777
EPZ005687
ERK5-IN-1
Esonarimod
ETC-159
Everolimus

F

FGF401
FICZ
Fluxametamide
Fumagillin

G

G-1
G-749
G007-LK
GANT 61
GDC-0152
GDC-0810
GDC-0994
Gdp 366
GGTI-2418
GLPG1690
Glutaminase C-IN-1
GM6001
GMB-475
GNE-140 racemate
GNE-493
GNE-495
GNE-6776
GPR84 Antagonist 8
GRA Ex-25
GSK 467
GSK'872
GSK-2018682
GSK1324726A
GSK2141795
GSK2193874
GSK2807 Trifluoroacetate
GSK429286A
GSK650394
GW2580
GW788388

H

H-D-Phe-Homopro-Arg-pNA Diacetate
HSP990
Hydroxyfasudil
Hydroxyhexamide

I

ICG 001
IDO-IN-2
INCB057643
IPI-549
IQ-1
Ispinesib
ITE
ITI-214

J

JG-98
JI-101
JNJ-17203212
JNJ-38877605
JNJ-42153605
JQEZ5

K

Ki16425
KN-93
KPT-276
KYA1797K

L

Lazertinib
Lersivirine
LOC14
LTURM 34
LY-2940094 Tartrate
LY-3000328
LY-3200882
LY2109761
LY2857785
LY2940680

M

M2I-1
MAT2A Inhibitor
MDL-29951
Merimepodib
Methyl 6-amino-6-deoxy-2,3-di-O-tetradecyl-?-D-glucopyranoside
MGCD-265
MI-136
Mivebresib
MK-4101
MK-8353
MK-8998
ML-18
ML-364
ML-390
MLi-2
MLN-4924
MOZ-IN-3

N

N'-(7-Fluoropyrrolo[1,2-a]quinoxalin-4-yl)pyrazine-2-carbohydrazide
N-((4,6-Dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-4-methyl-4'-(morpholinomethyl)-[1,1'-biphenyl]-3-carboxamide
N-((S)-1-Amino-3-(3-fluorophenyl)propan-2-yl)-5-chloro-4-(4-chloro-1-methyl-1H-pyrazol-5-yl)thiophene-2-carboxamide
N-((S)-1-Amino-3-(3-fluorophenyl)propan-2-yl)-5-chloro-4-(4-chloro-1-methyl-1H-pyrazol-5-yl)thiophene-2-carboxamide Hydrochloride
N-(3-((4aS,7aS)-2-Amino-4a,5,7,7a-tetrahydro-4H-furo[3,4-d][1,3]thiazin-7a-yl)-4-fluorophenyl)-5-fluoropicolinamide hydrochloride
N-(4-(1-Cyanocyclopentyl)phenyl)-2-((pyridin-4-ylmethyl)amino)nicotinamide Methanesulfonate
N-(4-Fluorobenzyl)-2-((R)-5-(3-methylureido)-2',4'-dioxo-2,3-dihydrospiro[indene-1,5'-oxazolidin]-3'-yl)-N-((S)-1,1,1-trifluoropropan-2-yl)acetamide
N-[4-(2-tert-Butylphenylsulfonyl)phenyl]-2,3,4-trihydroxy-5-(2-isopropylbenzyl)benzamide
Nadide
Naquotinib
NCGC00244536
NIBR-189
Nidufexor
NITD-349
NLG919
NMDAR antagonist 1
NVP-231
NVP-TNKS656

O

OAC1
Oclacitinib
OG-L002
Orexin 2 Receptor Agonist
OSI-027
OSI-930
OTSSP167

P

Pacritinib
PD1-PDL1 Inhibitor 1
PD1-PDL1 Inhibitor 2
Peramivir trihydrate
Peretinoin
Pexmetinib
PF-06282999
PF-3084014
PFK-158
PHA-848125
PI-3065
PKC412
PKI-587
PLX8394
Porcupine-IN-1
PP242
PT-2385
Pu-h 71
PZ-2891

Q

Quizartinib

R

R-268712
RAF265
Ramosetron Hydrochloride
Refametinib
RGX-104 Free Acid
RK-33
RMC-4550
RP-5264
RS-127445
Rs-504393

S

S-38093
S63845
Sabutoclax
SAG HCl
Savolitinib
SB-423562
SC75741
SCH-527123
SCH772984
SecinH3
SF-2523
SGX-523
SNX-2112
Solcitinib
SPHINX31
SR-18292
SR-4370
SR-9238
Staurosporine

T

TAK-243
TAK-659 Hydrochloride
TAS-103 dihydrochloride
TD-4208
Temsirolimus
Tenapanor
TG6-10-1
TH34
THZ531
TIC-10
TM5441
Topiroxostat
TP-0903
TPPU

t

trans-N1-(2-Phenylcyclopropyl)cyclohexane-1,4-diamine dihydrochloride

U

U-73122
UCPH-101

V

Vemurafenib
Ver-50589
Verdinexor
Verteporfin
VL-285
VLX1570
VX-11e
VX-765

W

Walrycin B
WNK463
WNT Agonist 1
Wp1130

X

XL413 xhydrochloride

Y

Y06036

Z

Zanubrutinib
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